| 货号 | 3934/50 |
| 别名 | (4R)-rel-1,4-Dihydro-2,6-dimethyl-4 |
| 是否允许进口 | 否 |
| 是否危险品 | 是 |
| 供应商 | Tocris |
| 生物活性 | Orally active antihypertensive agent which displays a wide range of activities in vitroandin vivo. Inhibits L-, N- and T-type Ca2+ channels. Also inhibits aldosterone-induced mineralocorticoid receptor activation. Exhibits cardioprotective and antiartherosclerotic effects. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 542.02 |
| 分子式 | C28H31N3O6 |
| 可溶性/溶解性 | Soluble to 75 mM in DMSO and to 10 mM in ethanol |
| 参考文献 | Kosakaet al (2010) The L-, N-, T-type triple calcium channel blocker benidipine acts as an antagonist of mineralocorticoid receptor, a member of nuclear receptor family. Eur.J.Pharmacol. 635 49. PMID: 20307534. Yaoet al (2006) Pharmacological, pharmacokinetic, and clinical properties of benidipine hydrochloride, a novel long-acting calcium channel blocker. J.Pharmacol.Sci. 100 243. PMID: 16565579. |