TC-G 1000 (50 MG)
货号：
5021/50 基本售价：
12274.1 元 规格：
50 mg
产品信息
概述| 货号 | 5021/50 |
| 别名 | 4-(6,7-Dihydro-1,3-dimethylbenzo[c]thien-4-yl)-1H-imidazole maleate |
性能| 供应商 | Tocris |
| 生物活性 | Potent and selective α2D-adrenoceptor agonist (Ki values are 8.6 pM and 110 nM for rat α2Dandα1 receptors respectively and 25, 26 and 100 nM for human α2A,α2Candα2B receptors respectively. Exhibits analgesic activity in a mouse model of abdominal irritation. Orally active. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 346.4 |
| 分子式 | C13H14N2S.C4 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| 参考文献 | Rosset al (2000) α2 adrenoceptor agonists as potential analgesic agents. 2. Discovery of 4-(4-Imidazo)-1,3-dimethyl-6,7-dihydrothianaphthene as a high-affinity ligand for the α2D adrenergic receptor. J.Med.Chem. 43 1423. PMID: 10715142. |
