LP 44 (50 MG)
货号：
2534/50 基本售价：
12274.1 元 规格：
50 mg
产品信息
概述| 货号 | 2534/50 |
| 别名 | 4-[2-(Methylthio)phenyl]-N-(1,2,3,4-tetrahydro-1-naphthalenyl)-1-piperazinehexanamidehydrochloride |
性能| 供应商 | Tocris |
| 生物活性 | High affinity 5-HT7 receptor agonist (Ki = 0.22 nM) that displays selectivity over 5-HT1A and 5-HT2A receptors (200- and > 1000-fold respectively). Induces relaxation of substance P-stimulated guinea pig ileum (EC50 = 2.56 μM). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 488.13 |
| 分子式 | C27H37N3OS.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 75 mM in ethanol |
| CAS号 | 824958-12-5 |
| 参考文献 | Leopoldoet al (2004) Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agents. J.Med.Chem. 47 6616. PMID: 15588097. |
