| 货号 | 1088/50 |
| 别名 | [S-(R*,R*)]-[3-[[1-(3,4-Dichlorophe |
| 供应商 | Tocris |
| 生物活性 | A potent, selective GABAB receptor antagonist (IC50 = 4 nM). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >96 % |
| 计算分子量 | 444.76 |
| 分子式 | C18H28Cl2NO3P.HCl |
| 可溶性/溶解性 | Soluble to 50 mM in DMSO and to 10 mM in ethanol with gentle warming |
| CAS号 | 149184-21-4 |
| 参考文献 | Kaupmannet al (1998) GABAB-receptor subtypes assemble into functional heteromeric complexes. Nature 396 683. PMID: 9872317. Froestlet al (1996) Potent, orally active GABAB receptor antagonists. Pharmacol.Rev.Comm. 8127. Bruggeret al (1993) The action of new potent GABAB receptor antagonists in the hemisected spinal cord preparation of the rat. Eur.J.Pharmacol. 235 153. PMID: 8390938. |