| 货号 | 1024/50 |
| 别名 | 1-[2-((3-Carbamoyl-4-hydroxy)phenox |
| 供应商 | Tocris |
| 生物活性 | Highly selective and potent β1-adrenoceptor antagonist (IC50 = 0.7 nM). Displays 10,000-fold selectivity over β2-adrenoceptors. Also available as part of the β-Adrenoceptor Antagonist Tocriset™. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >96 % |
| 计算分子量 | 567.39 |
| 分子式 | C23H25F3N4O5.2HCl |
| 可溶性/溶解性 | Soluble to 50 mM in water |
| CAS号 | 105737-62-0 |
| 参考文献 | Hiebleet al (1995) α-and β-adrenoceptors. From the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification. J.Med.Chem. 38 3415. PMID: 7658428. Kitagawaet al (1995) Determination of β-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective β-antagonists. Br.J.Pharmacol. 116 1635. PMID: 8564230. Dooleyet al (1986) CGP 20712A: a useful tool for quantitating β1- and β2-adrenoceptors. Eur.J.Pharmacol. 130 137. PMID: 2877892. |