TC-G 1001 (50 MG)
货号：
4879/50 基本售价：
11381.8 元 规格：
50 mg
产品信息
概述| 货号 | 4879/50 |
| 别名 | 4-[[2-[(2-Fluorophenyl)amino]-4-oxo-5(4H)-thiazolylidene]methyl]benzoic acid |
性能| 供应商 | Tocris |
| 生物活性 | GPR35 agonist (pEC50 values are 7.59 and 8.36 for β-arrestin and Gαq-i5Ca2+ assays respectively). Displays 1000-fold greater potency at human GPR35 receptors relative to mouse and rat GPR35 orthologs in an IP1 accumulation assay. More potent than zaprinast (Cat. No. 0947). |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 342.34 |
| 分子式 | C17H11FN2O3< |
| 可溶性/溶解性 | Soluble to 10 mM in DMSO |
| 参考文献 | Neetoo-Isseljeeet al (2013) High-throughput identification and characterization of novel, species-selective GPR35 agonists. J.Pharmacol.Exp.Ther. 344 568. PMID: 23262279. |
