LP 12 hydrochloride (50 MG)
货号:
2925/50 基本售价:
11381.8 元 规格:
50 mg
产品信息
概述货号 | 2925/50 |
别名 | 4-(2-Diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide hydrochloride |
性能供应商 | Tocris |
生物活性 | 5-HT7 receptor agonist displaying selectivity over D2, 5-HT1A and 5-HT2A receptors (Ki values are 0.22, 7.3, 52.7 and 326 nM respectively). Induces relaxation of substance P-induced contractions in guinea pig ileum (EC50 = 1.77 μM). |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >99 % |
计算分子量 | 518.13 |
分子式 | C32H39N30.HCl |
可溶性/溶解性 | Soluble to 75 mM in DMSO and to 75 mM in ethanol |
参考文献 | Leopoldoet al (2007) Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides, a class of 5-HT7 receptor agents. J.Med.Chem. 50 4214. PMID: 17649988. |