| 货号 | 1480/50 |
| 别名 | N-[1-[2-(4-Isothiocyanatophenyl)eth |
| 供应商 | Tocris |
| 生物活性 | Selective and irreversible δ-opioid agonist (EC50 = 8 nM); acts by alkylating the receptor. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >99 % |
| 计算分子量 | 393.55 |
| 分子式 | C23H27N3OS |
| 可溶性/溶解性 | Soluble to 100 mM in ethanol and to 10 mM in DMSO |
| CAS号 | 85951-63-9 |
| 参考文献 | Schoffelmeeret al (1988) μ-, δ- and κ-opioid receptor-mediated inhibition of neurotransmitter release and adenylate cyclase activity in rat brain slices: studies with fentanyl isothiocyanate. Eur.J.Pharmacol. 154 169. PMID: 2906610. Rothmanet al (1985) Evidence that the delta-selective alkylating agent, fit, alters the mu-noncompetitive opiate delta binding site. Neuropeptides 6 227. PMID: 2991807. Riceet al (1983) Irreversible ligands with high selectivity toward δ or μ opiate receptors. Science 220 314. PMID: 6132444. |