货号 | 2342/50 |
别名 | 5-(2-Aminoethyl)-4-methylimidazole dihydrochloride |
供应商 | Tocris |
生物活性 | Potent, high affinity H4 receptor agonist (Ki = 7 nM) that displays > 100-fold selectivity over other human histamine receptor subtypes. |
运输条件 | Blue Ice |
存放说明 | Ambient |
计算分子量 | 198.09 |
分子式 | C6H11N3.2HCl |
可溶性/溶解性 | Soluble to 50 mM in water |
CAS号 | 36376-47-3 |
参考文献 | Gbahouet al (2006) Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives. Br.J.Pharmacol 14774. Limet al (2005) Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist. J.Pharmacol.Exp.Ther. 314 1310. PMID: 15947036. |