DREADD agonist 21 (50 MG)
货号:
5548/50 基本售价:
11084.4 元 规格:
50 mg
产品信息
概述货号 | 5548/50 |
别名 | 11-(1-Piperazinyl)-5H-dibenzo[b,e][1,4]diazepine |
性能供应商 | Tocris |
生物活性 | Potent muscarinic hM3Dq DREADD agonist (EC50 = 1.7 nM). Highly selective for hM3Dq DREADDs over endogenous hM3receptors. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 278.35 |
分子式 | C17H18N4 |
可溶性/溶解性 | Soluble to 100 mM in DMSO and to 100 mM in ethanol |
参考文献 | Chenet al (2015) The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem.Neurosci. 18 476. PMID: 25587888. |