| 货号 | 3219/50 |
| 别名 | (3-Aminopropyl)ethylphosphinic acid hydrochloride |
| 供应商 | Tocris |
| 生物活性 | Selective GABAB antagonist. Displays activity at presynaptic receptors; ineffective at GABAB postsynaptic receptors. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 187.6 |
| 分子式 | C5H14NO2P.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in water and to 100 mM in DMSO |
| 参考文献 | Onget al (2001) CGP 36216 is a selective antagonist at GABAB presynaptic receptors in rat brain. Eur.J.Pharmacol. 415 191. PMID: 11274998. Froestlet al (1995) Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists. J.Med.Chem. 38 3313. PMID: 7650685. |