VU 152100 (50 MG)
货号：
3383/50 基本售价：
10489.5 元 规格：
50 mg
产品信息
概述| 货号 | 3383/50 |
| 别名 | 3-Amino-N-(4-methoxybenzyl)-4,6-dimethylthieno[2,3-b]pyridine carboxamide; ML 108 |
性能| 供应商 | Tocris |
| 生物活性 | Selective positive allosteric modulator of M4 muscarinic acetylcholine receptors (mAChRs) (EC50 = 380 nM). Induces 21-fold shift in ACh potency at M4 receptor. Displays no activity at other mAChR subtypes. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 341.43 |
| 分子式 | C18H19N3O2S |
| 可溶性/溶解性 | Soluble to 50 mM in DMSO |
| 参考文献 | Bradyet al (2008) Centrally active allosteric potentiators of the M4 muscarinic acetylcholine receptor reverse amphetamine-induced hyperlocomotor activity in rats. J.Pharmacol.Exp.Ther. 327 941. PMID: 18772318. |
