GSK 789472 hydrochloride (50 MG)
货号：
3940/50 基本售价：
9894.7 元 规格：
50 mg
产品信息
概述| 货号 | 3940/50 |
| 别名 | 4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one |
性能| 供应商 | Tocris |
| 生物活性 | Selective dopamine D3 receptor antagonist and D2 partial agonist (pEC50 values are <5.5 and 8.3 respectively). Selective against the D4 receptor in both agonist and antagonist assays. Brain penetrant. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 295.81 |
| 分子式 | C15H21N3O.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in water and to 100 mM in DMSO |
| 参考文献 | Holmeset al (2010) The identification of a selective dopamine D2 partial agonist, D3 antagonist displaying high levels of brain exposure. Bioorg.Med.Chem.Lett. 20 2013. PMID: 20153647. |
