| 货号 | 0914/50 |
| 别名 | (±)-1-[4-[[2-(1-Methylethoxy)ethoxy) |
| 供应商 | Tocris |
| 生物活性 | A selective β1-adrenergic antagonist. Has a Kd of 2-3 nM at the β1 receptor and a β1/β2 selectivity of approximately 100-fold. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 383.48 |
| 分子式 | C18H31NO4.紺4H4O4 |
| 可溶性/溶解性 | Soluble to 50 mM in water |
| CAS号 | 104344-23-2 |
| 参考文献 | Heibleet al (1995) α-and β-Adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification. J.Med.Chem. 38 3415. PMID: 7658428. Klockowet al (1986) Studies on the receptor profile of bisoprolol. Arzneimittelforschung 36 197. PMID: 2870719. Kaumann and Lemoine (1985) Direct labelling of myocardial β1-adrenoceptors. Comparison of binding affinity of 3H-(-)-bisoprolol with its blocking potency. Naunyn Schmiedebergs Arch.Pharmacol. 331 27. PMID: 2866449. |