| 货号 | 0892/50 |
| 别名 | 17-(Cyclopropylmethyl)-6,7-didehydr |
| 供应商 | Tocris |
| 生物活性 | Selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ,μandκ receptors respectively). Displays selectivity for the δ2subtypein vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 511.59 |
| 分子式 | C26H25NO4.CH3SO3H |
| 可溶性/溶解性 | Soluble to 50 mM in DMSO with gentle warming |
| CAS号 | 111555-58-9 |
| 参考文献 | Thorat and Hammond (1997) Modulation of nociception by microinjection of delta-1 and delta-2 opioid receptor ligands in the ventromedial medulla of the rat. J.Pharmacol.Exp.Ther. 283 1185. PMID: 9399992. Miyamotoet al (1993) Involvement of delta2 opioid receptors in the development of morphine dependence in mice. J.Pharmacol.Exp.Ther. 264 1141. PMID: 8383738. Portogheseet al (1991) Role of spacer and address components in peptidomimetic δ opioid receptor antagonists related to naltrindole. J.Med.Chem. 34 1715. PMID: 1851846. |