DY 268 (50 MG)
货号:
5656/50 基本售价:
9597.2 元 规格:
50 mg
产品信息
概述货号 | 5656/50 |
别名 | 1-[(3-Methoxyphenyl)methyl]-N-[4-methyl-3-(4-morpholinylsulfonyl)phenyl]-3-(4-methylphenyl)-1H-pyrazole-4-carboxamide |
性能供应商 | Tocris |
生物活性 | Potent FXR antagonist (IC50 = 7.5 nM). Exhibits no detectable cytotoxicity in cell-based assays. |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >98 % |
计算分子量 | 560.66 |
分子式 | C30H32N4O5 |
可溶性/溶解性 | Soluble to 100 mM in DMSO |
参考文献 | Yuet al (2014) Identification of trisubstituted-pyrazol carboxamide analogs as novel and potent antagonists of farnesoid X receptor. Bioorg.Med.Chem. 22 2919. PMID: 24775917. |