| 货号 | 0794/50 |
| 别名 | 2-(3,4-Dichlorophenyl)-N-methyl-N-[ |
| 供应商 | Tocris |
| 生物活性 | An irreversible and selective antagonist at the κ receptor, with persistent effect in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >99 % |
| 计算分子量 | 484.87 |
| 分子式 | C22H23Cl2N3OS.HCl |
| 可溶性/溶解性 | Soluble to 30 mM in ethanol and to 50 mM in DMSO |
| 参考文献 | Changet al (1994) 2-(3,4-Dichlorophenyl)-N-methyl-N-[(1S)-1-(3-isothiocyanatophenyl)-2-(1-pyrrolidinyl)ethyl]acetamide: an opioid receptor affinity label that produces selective and long lasting κ antagonism in mice. J.Med.Chem. 37 1547. PMID: 8201586. Changet al (1994) κ opioid receptor selective affinity labels: Electrophilic benzeneacetamides as κ-selective opioid antagonists. J.Med.Chem. 37 4490. PMID: 7799399. |