| 货号 | 1207/50 |
| 别名 | 3-[4-(4-Chlorophenyl)piperazin-1-yl |
| 供应商 | Tocris |
| 生物活性 | A selective h5-HT1D antagonist, displaying 60-fold selectivity over h5-HT1B, and exhibiting little or no affinity for a range of other receptor types. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 计算分子量 | 443.42 |
| 分子式 | C25H27ClN2O.HCl |
| 可溶性/溶解性 | Soluble to 10 mM in DMSO and to 50 mM in ethanol |
| CAS号 | 193611-72-2 |
| 参考文献 | Saxenaet al (1998) 5-HT1-like receptors: a time to bid goodbye. TiPS 19 311. PMID: 9745358. Haganet al (1997) Stimulation of 5-HT1B receptors causes hypothermia in the rat. Eur.J.Pharmacol. 331 169. PMID: 9274976. Priceet al (1997) SB-216641 and BRL-15572 - compounds to pharmacologically discriminate h5-HT1B and h5-HT1D receptors. Naunyn Schmiedebergs Arch.Pharmacol. 356 312. PMID: 9303567. Schlickeret al (1997) Effects of selective h5-HT1B (SB-216641) and h5-HT1D (BRL-15572) receptor ligands on guinea-pig and human 5-HT auto- and heteroreceptors. Naunyn Schmiedebergs Arch.Pharmacol. 356 321. PMID: 9303568. |