Perlapine (50 MG)
货号:
5549/50 基本售价:
9359.3 元 规格:
50 mg
产品信息
概述货号 | 5549/50 |
别名 | 6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine |
性能供应商 | Tocris |
生物活性 | Potent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). Exhibits >10,000-fold selectivity for hM3Dq over hM3. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >99 % |
计算分子量 | 291.39 |
分子式 | C19H21N3 |
可溶性/溶解性 | Soluble to 50 mM in DMSO and to 5 mM in water with gentle warming |
参考文献 | Chenet al (2015) The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem.Neurosci. 6 476. PMID: 25587888. |