| 货号 | 2021/50 |
| 别名 | 4-(7,8,9,10-Tetrahydro-5,7,7,10,10- |
| 供应商 | Tocris |
| 生物活性 | Retinoic acid antagonist; displays moderate selectivity for RARβ over RARα(Ki |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >97 % |
| 计算分子量 | 438.56 |
| 分子式 | C29H30N2O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| CAS号 | 155877-83-1 |
| 参考文献 | Liet al (1999) Identification of a novel class of retinoic acid receptor β-selective retinoid antagonists and their inhibitory effects on AP-1 activity and retinoic acid-induced apoptosis in human breast cancer cells. J.Biol.Chem. 274 15360. PMID: 10336422. Umemiyaet al (1997) Regulation of retinoidal actions by diazepinylbenzoic acids. Retinoid synergists which activate the RXR-RAR heterodimers. J.Med.Chem. 40 4222. PMID: 9435893. Eyrolleset al (1994) Retinobenzoic acids. 6. Retinoid antagonists with heterocyclic ring. J.Med.Chem. 37 1508. PMID: 8182710. |