JNJ 63533054 (50 MG)
货号：
5666/50 基本售价：
9359.3 元 规格：
50 mg
产品信息
概述| 货号 | 5666/50 |
| 别名 | 3-Chloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide |
性能| 供应商 | Tocris |
| 生物活性 | Potent and selective GPR139 agonist (EC50 = 16 nM). Selective for GPR139 over a panel of GPCRs, ion channels and transporters, including GPR142. Brain and cell penetrant. Orally bioavailable. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 316.78 |
| 分子式 | C17H17ClN2O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 20 mM in ethanol |
| 参考文献 | Dvoraket al (2015) Identification and SAR of glycine benzamides as potent agonists for the GPR139 receptor. ACS Med.Chem.Lett. 6 1015. PMID: 26396690. |
