| 货号 | 0347/50 |
| 别名 | 17,17'-(Dicyclopropylmethyl)-6,6',7,7 |
| 供应商 | Tocris |
| 生物活性 | A selective κ-opioid receptor antagonist. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 734.72 |
| 分子式 | C40H43N3O6.2HCl |
| 可溶性/溶解性 | Soluble to 25 mM in water with gentle warming and to 25 mM in DMSO |
| CAS号 | 105618-26-6 |
| 参考文献 | Blakeet al (1997) Differential agonist regulation of the human κ-opioid receptor. J.Neurochem. 68 1846. PMID: 9109509. Fenget al (1997) Nor-binaltorphimine precipitates withdrawal and excitatory amino acid release in the locus ceruleus of butorphanol- but not morphine-dependent rats. J.Pharmacol.Exp.Ther. 283 932. PMID: 9353416. Portogheseet al (1994) Structure-activity relationship of N17'-substituted norbinaltorphimine congeners. Role of the N17'-basic group in the interaction with a putative address subsite on the κ opioid receptor. J.Med.Chem. 37 1495. PMID: 8182708. |