| 货号 | 0778/50 |
| 别名 | 2-(3,4-Dichlorophenyl)-N-methyl-N-[ |
| 供应商 | Tocris |
| 生物活性 | Highly potent κ agonist, 146-fold more active than U-50488 (Cat. No. 0495) in vitro. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 427.8 |
| 分子式 | C21H24Cl2N2O.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 50 mM in ethanol |
| CAS号 | 115199-84-3 |
| 参考文献 | Barlowet al (1991) Structure/activity studies related to 2-(3,4-dichlorophenyl)-N-methyl-N-[2-(1-pyrrolidinyl)-1-substituted-ethyl]acetamides: a novel series of potent and selective κ-opioid agonists. J.Med.Chem. 34 3149. PMID: 1659636. Costelloet al (1991) 2-(3,4-Dichlorophenyl)-N-methyl-N-[2-(1-pyrrolidinyl)-1-substituted-ethyl]-acetamides: the use of conformational analysis in the development of a novel series of potent opioid κ agonists. J.Med.Chem. 34 181. PMID: 1846918. |