| 货号 | 1218/50 |
| 别名 | N-Pentanoyl-2-benzyltryptamine |
| 供应商 | Tocris |
| 生物活性 | A relatively potent MT2 melatonin receptor antagonist (pKi value = 8.03), displaying 89- and 229-fold selectivity over MT1 and GPR50 (melatonin-related orphan receptor) respectively. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 334.46 |
| 分子式 | C22H26N2O |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| 参考文献 | Tinget al (1999) Molecular and pharmacological evidence for MT1 melatonin receptor subtype in the tail artery of juvenile Wistar rats. Br.J.Pharmacol. 127 987. PMID: 10433507. Teh and Sugden (1998) Comparison of the relationships of melatonin receptor agonists and antagonists; lengthening the N-acyl side chain has differing effects on potency on Xenopus melanophores. Naunyn Schmiedebergs Arch.Pharmacol. 358 522. PMID: 9840420. |