货号 | 2698/1 |
别名 | Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide |
供应商 | Tocris |
生物活性 | Selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM for GAL2 and GAL1 receptors respectively). Blocks the pro-nociceptive effect of GAL2 receptor agonists. |
运输条件 | Blue Ice |
存放说明 | -20℃ |
计算分子量 | 2287.64 |
分子式 | C108H163N27O28 |
可溶性/溶解性 | Soluble to 1 mg/ml in 30% acetonitrile |
CAS号 | 908844-75-7 |
序列号 | WTLNSAGYLLGPEHPPPALALA (Modifications: Ala-22 = C-terminal amide) |
参考文献 | Jimenez-Andradeet al (2006) Activation of peripheral galanin receptors: differential effects on nociception. Pharmacol.Biochem.Behav. 85 273. PMID: 16996122. Sollenburget al (2006) M871 - a novel peptide antagonist selectively recognizing the galanin receptor type 2. Int.J.Pept.Res.Ther. 12115. |