WAY 207024 dihydrochloride (10 MG)
货号:
3890/10 基本售价:
3708.0 元 规格:
10 mg
产品信息
概述货号 | 3890/10 |
别名 | 6-[[4-[2-[4-(1,1-Dimethylethyl)phenyl]-1H-benzimidazol-7-yl]-i-piperazinyl]methyl]-quinoxaline dihydrochloride |
性能供应商 | Tocris |
生物活性 | Gonadotropin releasing hormone receptor (GnRH-R) antagonist. Exhibits potent affinity (IC50 values are 12 and 71 nM for human and rat GnRH receptors respectively). Lowers plasma leuteinizing hormone levels in the rat. Orally active. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >99 % |
计算分子量 | 549.54 |
分子式 | C30H32N6.2HCl |
可溶性/溶解性 | Soluble to 85 mM in DMSO |
参考文献 | Pelletieret al (2009) Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the gonadotropin releasing hormone receptor (GnRH-R). J.Med.Chem. 52 214. PMID: 19072222. |