WAY 207024 dihydrochloride (10 MG)
货号：
3890/10 基本售价：
3708.0 元 规格：
10 mg
产品信息
概述| 货号 | 3890/10 |
| 别名 | 6-[[4-[2-[4-(1,1-Dimethylethyl)phenyl]-1H-benzimidazol-7-yl]-i-piperazinyl]methyl]-quinoxaline dihydrochloride |
性能| 供应商 | Tocris |
| 生物活性 | Gonadotropin releasing hormone receptor (GnRH-R) antagonist. Exhibits potent affinity (IC50 values are 12 and 71 nM for human and rat GnRH receptors respectively). Lowers plasma leuteinizing hormone levels in the rat. Orally active. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 549.54 |
| 分子式 | C30H32N6.2HCl |
| 可溶性/溶解性 | Soluble to 85 mM in DMSO |
| 参考文献 | Pelletieret al (2009) Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the gonadotropin releasing hormone receptor (GnRH-R). J.Med.Chem. 52 214. PMID: 19072222. |
