| 货号 | 5992/1 |
| 供应商 | Tocris |
| 生物活性 | Potent apelin receptor antagonist (Ki = 82 nM; IC50 = 93 nM). Antagonizes the inhibitory affect of [Pyr1]-Apelin-13 on forskolin-induced cAMP accumulation in CHO-K1-APJ cells. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 1737.15 |
| 分子式 | C70H121N29O1 |
| 可溶性/溶解性 | Soluble to 2 mg/ml in water |
| 序列号 | CRPRLCKHCRPRLC (Modifications: Disulfide bridge: 1-6,9-14) |
| 参考文献 | Macalusoet al (2011) Discovery of a competitive apelin receptor (APJ) antagonist. ChemMedChem 6 1017. PMID: 21560248. |