(1R,1S,3R/1R,1R,3S)-L-054,264 (10 MG)
货号:
2444/10 基本售价:
3648.5 元 规格:
10 mg
产品信息
概述货号 | 2444/10 |
别名 | N-[(1R)-2-[[[(1S*,3R*)-3-(Aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]spiro[1H-indene-1,4'-piperidine]-1'-carboxamide |
性能供应商 | Tocris |
生物活性 | Potent and selective somatostatin sst2 receptor agonist (Ki values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst2, sst1, sst4, sst3 and sst5 receptors respectively). |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >96 % |
计算分子量 | 539.71 |
分子式 | C33H41N5O2 |
可溶性/溶解性 | Soluble to 50 mM in DMSO and to 100 mM in ethanol |
CAS号 | 208706-12-1 |
参考文献 | Yanget al (1998) Spiro[1H-indene-1,4'-piperidine] derivatives as potent and selective non-peptide human somatostatin receptor subtype 2 (sst2) agonists. J.Med.Chem. 41 2175. PMID: 9632348. |