货号 | 1688/1 |
别名 | AIP |
供应商 | Tocris |
生物活性 | Selective and potent calmodulin-dependent protein kinase II (CaM kinase II) inhibitor (IC50 = 40 nM). Selective over PKC, PKA and CaM kinase IV (IC50 > 10 μM). |
运输条件 | Blue Ice |
存放说明 | -20℃ |
计算分子量 | 1497.76 |
分子式 | C64H116N22O19 |
可溶性/溶解性 | Soluble to 1 mg/ml in water |
CAS号 | 167114-91-2 |
序列号 | KKALRRQEAVDAL |
参考文献 | Ishidaet al (1995) A novel highly specific and potent inhibitor of calmodulin-dependent protein kinase II. Biochem.Biophys.Res.Commun. 212 806. PMID: 7626114. Ishida and Fujisawa (1995) Stabilization of calmodulin-dependent protein kinase II through the autoinhibitory domain. J.Biol.Chem. 270 2163. PMID: 7836445. Takasawaet al (1995) Requirement of calmodulin-dependent protein kinase II in cyclic ADP-ribose-mediated intracellular Ca2+ mobilization. J.Biol.Chem. 270 30257. PMID: 8530441. |