货号 | 3007/1 |
供应商 | Tocris |
生物活性 | Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94). |
运输条件 | Blue Ice |
存放说明 | -20℃ |
计算分子量 | 2138.56 |
分子式 | C96H156N34O20S |
可溶性/溶解性 | Soluble to 1.20 mg/ml in water |
CAS号 | 217082-57-0 |
序列号 | KFRRQRPRLSHKGPMPF |
参考文献 | De Motaet al (2004) Apelin, a potent diuretic neuropeptide counteracting vasopressin actions through inhibition of vasopressin neuron activity and vasopressin release. Proc.Natl.Acad.Sci. USA 10110464. Medhurstet al (2003) Pharmacological and immunohistochemical characterization of the APJ receptor and its endogenous ligand apelin. J.Neurochem. 84 1162. PMID: 12603839. Tatemotoet al (1998) Isolation and characterization of a novel endogenous peptide ligand for the human APJ receptor. Biochem.Biophys.Res.Comms. 251471. |