| 货号 | 2207/1 |
| 供应商 | Tocris |
| 生物活性 | Novel cyclic peptide that disrupts interaction between GluR6 and the postsynaptic density protein 95 (PSD-95). Competes with the C-terminus of GluR6 for binding to the PDZ1 domain of PSD-95. Inhibits clustering of kainate receptors. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 819.95 |
| 分子式 | C38H61N9O11 |
| 可溶性/溶解性 | Soluble to 1 mg/ml in 5% acetonitrile / water and to 4 mg/ml in DMSO |
| 序列号 | YKKTEAV (Modifications: Ala-6 = β-Ala, Cyclized = Lys-3 - Ala-6)) |
| 参考文献 | Piserchioet al (2004) Targeting specific PDZ domains of PSD-95: structural basis for enhanced affinity and enzymatic stability of a cyclic peptide. Chem.Biol. 11 469. PMID: 15123241. |