| 货号 | 1836/1 |
| 别名 | MK 678 |
| 供应商 | Tocris |
| 生物活性 | Peptide agonist for sst2 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: > 1000 (sst1), 0.2 - 1.5 (sst2), 27 - 36 (sst3), > 127 (sst4), and 0.06 - 23 (sst5). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 808.98 |
| 分子式 | C44H56N8O7 |
| 可溶性/溶解性 | Soluble to 1 mg/ml in water |
| CAS号 | 81377-02-8 |
| 序列号 | AYWKVF (Modifications: Ala-1 = N-methyl-Ala, Trp-3 = D-Trp, Cyclized) |
| 参考文献 | Hannonet al (2002) Drug design at peptide receptors. Somatostatin receptor ligands. J.Mol.Neurosci. 1815. Hoyeret al (1994) Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch.Pharmacol. 350 441. PMID: 7870182. Raynoret al (1993) Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding to linear peptides. Mol.Pharmacol. 43 838. PMID: 8100350. |