| 货号 | 3935/10 |
| 别名 | 5-(6,7-Dihydrobenzo[b]thien-4-yl-1H |
| 供应商 | Tocris |
| 生物活性 | Agonist of the α2D adrenergic receptor (Ki values are 1.5, 254, 443 and 621 nM for α2D,α2A,α1 and α2B adrenergic receptors respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 202.28 |
| 分子式 | C11H10N2S |
| 可溶性/溶解性 | Soluble to 50 mM in DMSO and to 50 mM in ethanol |
| 参考文献 | Amphouxet al (2010) Inhibitory and facilitatory actions of isocyanine derivatives at human and rat organic cation transporters 1, 2 and 3: a comparison to human α1- and α2-adrenoceptor subtypes. Eur.J.Pharmacol. 634 1. PMID: 20170649. Rosset al (2000) α2 adrenoceptor agonists as potential analgesic agents. 2. Discovery of 4-(4-imidazo)-1,3-dimethyl-6,7-dihydrothianaphthene as a high-affinity ligand for the α2D adrenergic receptor. J.Med.Chem. 43 765. PMID: 10753480. |