| 货号 | 1904/1 |
| 供应商 | Tocris |
| 生物活性 | Potent inhibitor of cAMP-dependent protein kinase (PKA) (Ki = 2.5 nM); derived from the active portion of the heat-stable PKA inhibitor protein PKI. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 1868.08 |
| 分子式 | C80H130N28O24 |
| 可溶性/溶解性 | Soluble to 1 mg/ml in water |
| CAS号 | 121932-06-7 |
| 序列号 | TYADFIASGRTGRRNAI (Modifications: Ile-17 = C-terminal amide) |
| 参考文献 | Otmakhovaet al (2000) Inhibition of the cAMP pathway decreases early long-term potentiation at CA1 hippocampal synapses. J.Neurosci. 20 4446. PMID: 10844013. Glasset al (1989) Primary structural determinants essential for potent inhibition of cAMP-dependent protein kinase by inhibitory peptides corresponding to the active portion of the heat-stable inhibitor protein. J.Biol.Chem. 264 8802. PMID: 2722799. Glasset al (1989) Protein kinase inhibitor-(6-22)-amide peptide analogs with standard and nonstandard amino acid substitutions for phenylalanine 10. J.Biol.Chem. 264 14579. PMID: 2760075. |