| 货号 | 0234/100 |
| 别名 | 1,2,5,6-Tetrahydropyridine-3-carbox |
| 供应商 | Tocris |
| 生物活性 | Specific GABA uptake inhibitor. IC50 values are 14, 58, 119 and 1870 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 163.6 |
| 分子式 | C6H9NO2.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in water |
| CAS号 | 498-96-4 |
| 参考文献 | Bordenet al (1994) Tiagabine, SK&F 89976-A, CI 966, and NNC-711 are selective for the cloned GABA transporter GAT-1. Eur.J.Pharmacol. 269 219. PMID: 7851497. Krogsgaard-Larsenet al (1978) Structure-activity studies on the inhibition of GABA binding to rat brain membranes by muscimol and related compounds. J.Neurochem. 30 1377. PMID: 670980. |