| 货号 | 1387/1 |
| 供应商 | Tocris |
| 生物活性 | Potent, selective partial agonist peptide for the NOP receptor (Ki = 0.71 nM). Selective over μ,δandκ opioid receptors (IC50 > 4000 nM). Increases food intake in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 1012.17 |
| 分子式 | C49H69N15O9 |
| 可溶性/溶解性 | Soluble to 1 mg/ml in water |
| CAS号 | 200959-47-3 |
| 序列号 | RYYRWK (Modifications: Arg-1 = C-terminal Ac, Lys-6 = C-terminal amide) |
| 参考文献 | Hoet al (2000) Characterization of the ORL1 receptor on adrenergic nerve in the rat anococcygeus. Br.J.Pharmacol. 131 349. PMID: 10991930. Dooleyet al (1997) Binding and in vitro activities of peptides with high affinity for the nociceptin/orphanin FQ receptor, ORL1. J.Pharmacol.Exp.Ther. 283 735. PMID: 9353393. |