货号 | 3138/50U |
别名 | 4-[[(1R,2E,4E,6Z,9Z)-1-[(1S)-4-Carb |
供应商 | Tocris |
生物活性 | Cysteinyl leukotriene receptor antagonist with equal affinity at both CysLT1 and CysLT2 receptors (pKB values are 6.8 and 6.5 respectively). Competitive antagonist of LTC4- and LTE4-induced contractions of the guinea pig trachea. |
运输条件 | Dry Ice |
存放说明 | -80℃ |
计算分子量 | 472.64 |
分子式 | C27H36O5S |
可溶性/溶解性 | Soluble in ethanol (supplied pre-dissolved in Ethanol, 0.1mg/ml) |
参考文献 | Back (2002) Functional characteristics of cysteinyl-leukotriene receptor subtypes. Life Sci. 71 611. PMID: 12072150. Goranneet al (1996) Cysteinyl leukotriene receptors in the human lung: what's new? TiPS 17 342. PMID: 8979767. Labatet al (1992) A second cysteinyl leukotriene receptor in human lung. J.Pharmacol.Exp.Ther. 263 800. PMID: 1331415. |