| 货号 | 2403/10 |
| 别名 | 2-Phenoxy-6-(cyclohexylamino)purine |
| 供应商 | Tocris |
| 生物活性 | High affinity adenosine A3 receptor antagonist (Ki = 47 nM) that displays > 200-fold selectivity versus A1, A2A and A2Breceptors. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 354.39 |
| 分子式 | C17H19N5O.紺2H2O4 |
| 可溶性/溶解性 | Soluble to 50 mM in DMSO |
| 参考文献 | Jacobson and Gao (2006) Adenosine receptors as therapeutic targets. Nat.Rev.Drug Discov. 5 247. PMID: 16518376. Moroet al (2006) Progress in the pursuit of therapeutic adenosine receptor antagonists. Med.Res.Rev. 26 131. PMID: 16380972. Perreiraet al (2005) "Reversine" and its 2-substituted adenine derivatives as potent and selective A3 adenosine receptor antagonists. J.Med.Chem. 48 4910. PMID: 16033270. |