| 货号 | 4588/10 |
| 别名 | 2,2',2'',2'''-[[4,8-Bis(hexahydro-1(2H)-a |
| 供应商 | Tocris |
| 生物活性 | Potent equilibrative nucleoside transporter 1 (ENT1) inhibitor (IC50 = 0.43 nM). Inhibits hENT1 and hENT2 uptake of [H3]uridine in K562 cells and K15NTD cells respectively. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >98 % |
| 计算分子量 | 560.73 |
| 分子式 | C28H48N8O4 |
| 可溶性/溶解性 | Soluble to 20 mM in DMSO |
| 参考文献 | Linet al (2011) Design, synthesis, and evaluation of 2-diethanolamino-4,8-diheptamethyleneimino-2-(N-aminoethyl-N-ethanolamino)-6-(N,N-diethanolamino)pyrimido[5,4-d]pyrimidine-fluorescein conjugate (8MDP-fluor), as a novel equilibrative nucleoside transporter probe. Bioconjug.Chem. 22 1221. PMID: 21539390. Linet al (2007) Synthesis, flow cytometric evaluation, and identification of highly potent dipyridamole analogues as equilibrative nucleoside transporter 1 inhibitors. J.Med.Chem. 50 3906. PMID: 17636949. |