货号 | 1860/10 |
别名 | 1-(2,3-Dihydro-1,4-benzodioxin-5-yl |
供应商 | Tocris |
生物活性 | 5-HT1 and 5-HT2C receptor partial agonist (Ki values are 40, 52 and 81 nM for 5-HT1A, 5-HT1B and 5-HT2C receptors respectively). Reduces 5-HIAA levels in the striatum and exhibits antiaggressive behavior in vivo. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 256.73 |
分子式 | C12H16N2O2 |
可溶性/溶解性 | Soluble to 100 mM in water |
参考文献 | Gommanset al (1997) Discriminative stimulus properties of eltoprazine. Life Sci. 61 11. PMID: 9200664. Schipperet al (1990) Neurochemical profile of eltoprazine. Drug Metabol.Drug Interact. 8 85. PMID: 1982626. Miczeket al (1989) Brain 5-HT and inhibition of aggressive behavior in animals: 5-HIAA and receptor subtypes. Psychopharmacol.Bull. 25 399. PMID: 2483273. |