货号 | 1506/50 |
别名 | 1-(4-Amino-6,7-dimethoxy-2-quinazol |
供应商 | Tocris |
生物活性 | α1- and α2B-adrenoceptor antagonist (Ki values are 3.3, 0.7, 1.1, 7.7, 1510 and 78.2 nM for α1A,α1B,α1D,α2B,α2Aandα2C receptors respectively). Antihypertensive following oral or intravenous administration in vivo. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >99 % |
计算分子量 | 423.9 |
分子式 | C19H25N5O4.HCl |
可溶性/溶解性 | Soluble to 50 mM in water with gentle warming |
CAS号 | 63074-08-8 |
参考文献 | Hancocket al (1995) Actions of terazosin and its enantiomers at subtypes of α1- and α2-adrenoceptors in vitro. J.Recept.Signal Transduct.Res. 15 863. PMID: 8673721. Maruyamaet al (1994) Comparison of displacemental potencies of terazosin enantiomers for α1-adrenoceptor subtypes. Biol.Pharm.Bull. 17 1126. PMID: 7820122. Kyncl (1986) Pharmacology of terazosin. Am.J.Med. 80 12. PMID: 2872801. |