| 货号 | 1056/5 |
| 供应商 | Tocris |
| 生物活性 | Endogenous peptide with extremely high affinity and selectivity for μ-opioid receptors (with Ki values of 0.69, 9233 and 5240 nM for μ,δandκrespectively). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 571.65 |
| 分子式 | C32H37N5O5 |
| 可溶性/溶解性 | Soluble to 0.40 mg/ml in water |
| CAS号 | 141801-26-5 |
| 序列号 | YPFF (Modifications: Phe-3 = C-terminal amide) |
| 参考文献 | Goldberget al (1998) Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J.Pharmacol.Exp.Ther. 286 1007. PMID: 9694962. Harrisonet al (1998) Differential effects of endomorphin-1, endomorphin-2, and tyr-W-MIF-1 on activation of G-proteins in SH-SY5Y human neuroblastoma membranes. Peptides 19 749. PMID: 9622031. Chapmanet al (1997) Distinct inhibitory effects of spinal endomorphin-1 and endomorphin-2 on evoked dorsal horn neuronal responses in the rat. Br.J.Pharmacol. 122 1537. PMID: 9422796. Zadinaet al (1997) A potent and selective endogenous agonist for the μ-opiate receptor. Nature 386 499. PMID: 9087409. |