| 货号 | 1055/5 |
| 供应商 | Tocris |
| 生物活性 | Endogenous peptide with an exceptionally high affinity (Ki = 360 pM) and selectivity for μ opioid receptors (4000- and 15000-fold preference over δandκrespectively). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 610.67 |
| 分子式 | C34H38N6O5 |
| 可溶性/溶解性 | Soluble to 0.60 mg/ml in water |
| CAS号 | 189388-22-5 |
| 序列号 | YPWF (Modifications: Phe-3 = C-terminal amide) |
| 参考文献 | Goldberget al (1998) Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J.Pharmacol.Exp.Ther. 286 1007. PMID: 9694962. Harrisonet al (1998) Differential effects of endomorphin-1, endomorphin-2, and tyr-W-MIF-1 on activation of G-proteins in SH-SY5Y human neuroblastoma membranes. Peptides 19 749. PMID: 9622031. Kakizawaet al (1998) Parallel stimulations of in vitro and in situ [35S]GTPγS binding by endomorphin 1 and DAMGO in mouse brains. Peptides 19 755. PMID: 9622032. Zadinaet al (1997) A potent and selective endogenous agonist for the μ-opiate receptor. Nature 386 499. PMID: 9087409. |