Taranabant
货号：
10009795-5mg 基本售价：
3920.0 元 规格：
5 mg
产品信息
概述| 货号 | 10009795-5mg |
| 描述 | Taranabant is an inverse agonist at the central cannabinoid (CB) receptor CB1(IC50 = 35 nM for rat brain CB1).1 It has little effect at human CB2(IC50 > 10 µM).1 In a published study, taranabant mediated weight loss by increasing energy expenditure and decreasing caloric intake.2 |
| 别名 | MK-0364; |
性能| 供应商 | Cayman |
| 应用文献 |
1.Lee, S.H.,Seo, H.J.,Lee, S.H., et al. Biarylpyrazolyl oxadiazole as potent, selective, orally bioavailable cannabinoid-1 receptor antagonists for the treatment of obesity. J. med. Chem. 51, 7216-7233 (2008).
2.Addy, C.,Wright, H.,Van Laere, K., et al. The acyclic CB1R inverse agonist taranabant mediates weight loss by increasing energy expenditure and decreasing caloric intake. Cell Metab. 7, 68-78 (2008).
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| 运输条件 | Room temperature in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 516 |
| 分子式 | C27H25ClF3N3O2 |
| CAS号 | 701977-09-5 |
| 稳定性 | ≥ 2 years |
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